COMPOUNDS / GABAERGIC / KAVA
GABAERGIC

KAVA

MEDIUM RISK
BEST FOR:Anxiety●●●●●●●○○○7/10
KAVA · PIPER METHYSTICUM · KAVA-KAVA · KAVAKAVA · KAVA ROOT · KAVALACTONE · AWA · AVA · YAQONA · SAKAU · RAUSCHPFEFFER · KAVA PEPPER
AnxiolyticGABAergicPacific IslanderHerbal SupplementSedativeTraditional Medicine

Traditional Pacific Islander root beverage with anxiolytic and sedative effects from kavalactones, used for centuries in ceremonial and social contexts.

ROUTE / DOSAGE
LOW60mg
STANDARD120-280mg
HIGH400mg+
Note: Dose refers to kavalactone content; traditional root preparation may require 10-30g root powder to achieve equivalent kavalactone dose
CYCLE
Daily use up to 4-8 weeks take breaks to reduce tolerance and hepatotoxicity risk
BIOAVAILABILITY
~20-40% oral higher with traditional lipid-rich preparation
ACTIVE DURATION
4-8h (subjective)
STORAGE
Room temperature dry away from light prepared beverage should be consumed fresh
HALF-LIFE
~9h (plasma)
DURATION BREAKDOWN
Total4-8h
Onset20-45min
Come up30-60min
Peak1-3h
Offset2-4h
After effects2-6h
Duration varies by route, dose, and individual. Source: community reports.
§ 01 — EFFECTS
8 documented
Anxiolysis and stress relief
Muscle relaxation
Mild sedation
Sociability enhancement
Mild euphoria
Numbing of mouth and throat
Improved sleep quality
Maintained mental clarity
§ 02 — RISKS
Rare but serious hepatotoxicity including hepatitis and liver failure, mechanism poorly understood
Reversible dermopathy (dry, scaly skin) with prolonged heavy use
Potential for dependence and withdrawal syndrome with heavy chronic use including delirium and sympathetic activation
Hyponatremia and altered mental status reported with heavy intoxication
Drug interactions with other CNS depressants, alcohol, and CYP substrates
Potential contamination or lack of standardization across products
§ 03 — INTERACTIONS
No interaction with your stack
VIEW STACK
CAUTION
Stimulants
AVOID · DANGEROUS
Depressants
Dissociatives
§ 04 — SCIENCE

Multiple randomized placebo-controlled trials support kava extract as superior to placebo for generalized anxiety disorder, with effect sizes of 0.59-0.99 in meta-analyses. Short-term use (4-8 weeks) at 120-280mg kavalactones daily is generally well tolerated with mild, transient adverse events. However, rare but serious hepatotoxicity has been reported, leading to regulatory restrictions in several countries; the mechanism remains unclear and may relate to non-kavalactone constituents or specific extract preparations. Evidence for anti-inflammatory and anticancer effects is preliminary and based largely on preclinical data. Long-term safety data are insufficient, and product standardization remains a significant challenge.

§ 06 — SOURCES
[1]
Kava as a Clinical Nutrient: Promises and Challenges
pubmed.ncbi.nlm.nih.gov ↗
[2]
Kava Withdrawal Treated With Phenobarbital - A Case Report and Literature Review
pubmed.ncbi.nlm.nih.gov ↗
[3]
Kava for Generalized Anxiety Disorder: A Review of Current Evidence
pubmed.ncbi.nlm.nih.gov ↗
[4]
Kava: An Overview
pubmed.ncbi.nlm.nih.gov ↗
[5]
Kava-kava and Anxiety: Growing Knowledge About Efficacy and Safety
pubmed.ncbi.nlm.nih.gov ↗
[6]
Toxicity of Kava Kava
pubmed.ncbi.nlm.nih.gov ↗
[7]
Kava Extract for Treating Anxiety (Cochrane Review)
pubmed.ncbi.nlm.nih.gov ↗
[8]
Kava Consumption and Its Health Effects
pubmed.ncbi.nlm.nih.gov ↗
[9]
PsychonautWiki - Kava
psychonautwiki.org ↗
Disclaimer. Protokol.wiki is an informational reference. Nothing on this site is medical advice. Compounds listed may be unapproved, unregulated, or illegal in your jurisdiction. Consult a licensed physician before use. Data compiled from peer-reviewed literature.
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