COMPOUNDS / / CREATINE

CREATINE

LOW RISK

Naturally occurring compound that increases cellular phosphocreatine stores, enhancing ATP regeneration for muscle and brain energy metabolism.

ROUTE / DOSAGE
LOW3g
STANDARD5g
HIGH20g
CYCLE
Daily use acceptable optional loading phase 20g/day for 5-7 days then 3-5g/day maintenance
BIOAVAILABILITY
—
ACTIVE DURATION
—
STORAGE
—
HALF-LIFE
~3h (plasma)
§ 01 — EFFECTS
6 documented
Increased muscle phosphocreatine stores
Improved performance in short-duration high-intensity exercise
Enhanced recovery between training bouts
Increased lean body mass via intracellular water retention
Potential cognitive benefits during metabolic stress
Possible mood improvement and antidepressant effects
§ 02 — RISKS
Weight gain from intracellular water retention (typically 1-2 kg)
Gastrointestinal discomfort at higher doses
Theoretical renal stress in individuals with pre-existing kidney disease
Lack of long-term safety data in children and adolescents
Possible increased hair loss or baldness (evidence weak and conflicting)
Product contamination or adulteration in unregulated supplement markets
§ 03 — INTERACTIONS
Interaction data not yet available for this compound.
§ 04 — SCIENCE

Over 500 peer-reviewed studies support creatine monohydrate as an effective ergogenic aid for short-duration, high-intensity exercise, with recommended dosages of 3-5 g/day or 0.1 g/kg body mass/day showing consistent benefits in muscle performance and recovery. Emerging research suggests creatine supplementation can increase brain creatine stores, with preliminary evidence for improved cognition during sleep deprivation, attenuation of concussion symptoms, and modest antidepressant effects. Evidence for neurodegenerative disease applications (e.g., multiple sclerosis) remains limited and inconclusive. Short-term use is generally well tolerated, though long-term safety data in children and adolescents is lacking. Many study authors have industry ties to creatine manufacturers, which warrants consideration when interpreting the evidence base.

§ 06 — SOURCES
[1]
Common questions and misconceptions about creatine supplementation: what does the scientific evidence really show?
pubmed.ncbi.nlm.nih.gov ↗
[2]
Effects of Creatine Supplementation on Brain Function and Health
pubmed.ncbi.nlm.nih.gov ↗
[3]
Creatine in Health and Disease
pubmed.ncbi.nlm.nih.gov ↗
[4]
Creatine Use in Sports
pubmed.ncbi.nlm.nih.gov ↗
[5]
Creatine in women's health: bridging the gap from menstruation through pregnancy to menopause
pubmed.ncbi.nlm.nih.gov ↗
[6]
Creatine and multiple sclerosis
pubmed.ncbi.nlm.nih.gov ↗
[7]
Heads Up for Creatine Supplementation and its Potential Applications for Brain Health and Function
pubmed.ncbi.nlm.nih.gov ↗
[8]
PsychonautWiki - Creatine
psychonautwiki.org ↗
Disclaimer. Protokol.wiki is an informational reference. Nothing on this site is medical advice. Compounds listed may be unapproved, unregulated, or illegal in your jurisdiction. Consult a licensed physician before use. Data compiled from peer-reviewed literature.
METHODOLOGYCONTRIBUTECONTACT